Comparison of different methods for estimation of lipophilicity of propafenone-type modulators of multidrug resistance

Author(s)
S. Prets, A. Jungreithmair, P. Chiba, G. Ecker
Abstract

Lipophilicity values of a series of 23 propafenone-type MDR-modulators were estimated using various software packages and compared with lipophilicity indices obtained by an HPLC method. Best correlations were obtained for MOLGEN® (r = 0.990) and the spl-macro 'logP' from SYBYL® (r = 0.980).

Organisation(s)
External organisation(s)
University of Vienna
Journal
Scientia Pharmaceutica
Volume
64
Pages
627-636
No. of pages
10
ISSN
0036-8709
Publication date
09-1996
Peer reviewed
Yes
Austrian Fields of Science 2012
301207 Pharmaceutical chemistry
Keywords
ASJC Scopus subject areas
Pharmaceutical Science
Portal url
https://ucrisportal.univie.ac.at/en/publications/080ed009-987c-426f-b432-ebe03ce9637b