Publications, Patents, Books and Book Chapters
Showing entries 71 - 80 out of 260
2017
Sanz, F, Pognan, F, Steger-Hartmann, T, Díaz, C, Cases, M, Pastor, M, Marc, P, Wichard, J, Briggs, K, Watson, DK, Kleinöder, T, Yang, C, Amberg, A, Beaumont, M, Brookes, AJ, Brunak, S, Cronin, MTD, Ecker, GF, Escher, S, Greene, N, Guzmán, A, Hersey, A, Jacques, P, Lammens, L, Mestres, J, Muster, W, Northeved, H, Pinches, M, Saiz, J, Sajot, N, Valencia, A, van der Lei, J, Vermeulen, NPE, Vock, E, Wolber, G & Zamora, I 2017, 'Legacy data sharing to improve drug safety assessment: the eTOX project', Nature Reviews. Drug Discovery, vol. 16, no. 12, pp. 811-812. https://doi.org/10.1038/nrd.2017.177
Jorgensen, L, Al-Khawaja, A, Kickinger, S, Vogensen, SB, Skovgaard-Petersen, J, Rosenthal, E, Borkar, N, Loffler, R, Madsen, KK, Brauner-Osbome, H, Schousboe, A, Ecker, GF, Wellendorph, P & Causen, RP 2017, 'Structure-Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/γ-Aminobutyric Acid Transporter 1 (BGT1)', Journal of Medicinal Chemistry, vol. 60, no. 21, pp. 8834-8846. https://doi.org/10.1021/acs.jmedchem.7b00924
Leist, M, Ghallab, A, Graepel, R, Marchan, R, Hassan, R, Bennekou, SH, Limonciel, A, Vinken, M, Schildknecht, S, Waldmann, T, Danen, E, van Ravenzwaay, B, Kamp, H, Gardner, I, Godoy, P, Bois, FY, Braeuning, A, Reif, R, Oesch, F, Drasdo, D, Höhme, S, Schwarz, M, Hartung, T, Braunbeck, T, Beltman, J, Vrieling, H, Sanz, F, Forsby, A, Gadaleta, D, Fisher, C, Kelm, J, Fluri, D, Ecker, G, Zdrazil, B, Terron, A, Jennings, P, van der Burg, B, Dooley, S, Meijer, AH, Willighagen, E, Martens, M, Evelo, C, Mombelli, E, Taboureau, O, Mantovani, A, Hardy, B, Koch, B, Escher, S, van Thriel, C, Cadenas, C, Kroese, D, van de Water, B & Hengstler, JG 2017, 'Adverse outcome pathways: opportunities, limitations and open questions', Archives of Toxicology, vol. 91, no. 11, pp. 3477–3505. https://doi.org/10.1007/s00204-017-2045-3
Damgaard, M, Haugaard, AS, Kickinger, S, Al-Khawaja, A, Lie, MEK, Ecker, G, Clausen, RP & Frølund, B 2017, Development of Non-GAT1-Selective Inhibitors: Challenges and Achievements. in A Ortega & A Schousboe (eds), Glial Amino Acid Transporters. Springer, Advances in Neurobiology.
Kotsampasakou, E, Montanari, F & Ecker, GF 2017, 'Predicting drug-induced liver injury: The importance of data curation', Toxicology, vol. 389, pp. 139-145. https://doi.org/10.1016/j.tox.2017.06.003
Spork, M, Sohail, MI, Schmid, D, Ecker, GF, Freissmuth, M, Chiba, P & Stockner, T 2017, 'Folding correction of ABC-transporter ABCB1 by pharmacological chaperones: a mechanistic concept', Pharmacology Research & Perspectives, vol. 5, no. 3, e00325, pp. e00325. https://doi.org/10.1002/prp2.325
Schuetz, DA, de Witte, WEA, Wong, YC, Knasmueller, B, Richter, L, Kokh, DB, Sadiq, SK, Bosma, R, Nederpelt, I, Heitman, LH, Segala, E, Amaral, M, Guo, D, Andres, D, Georgi, V, Stoddart, LA, Hill, S, Cooke, RM, De Graaf, C, Leurs, R, Frech, M, Wade, RC, de Lange, ECM, IJzerman, AP, Müller-Fahrnow, A & Ecker, GF 2017, 'Kinetics for Drug Discovery: an industry-driven effort to target drug residence time', Drug Discovery Today, vol. 22, no. 6, pp. 896-911. https://doi.org/10.1016/j.drudis.2017.02.002
Jain, S, Grandits, M, Richter, L & Ecker, GF 2017, 'Structure based classification for bile salt export pump (BSEP) inhibitors using comparative structural modeling of human BSEP', Journal of Computer-Aided Molecular Design, vol. 31, no. 6, pp. 507-521. https://doi.org/10.1007/s10822-017-0021-x
Seddik, A, Geerke, DP, Stockner, T, Holy, M, Kudlacek, O, Cozzi, NV, Ruoho, AE, Sitte, HH & Ecker, GF 2017, 'Combined Simulation and Mutation Studies to Elucidate Selectivity of Unsubstituted Amphetamine-like Cathinones at the Dopamine Transporter', Molecular Informatics, vol. 36, no. 5-6, 1600094. https://doi.org/10.1002/minf.201600094
Kotsampasakou, E, Escher, SE & Ecker, GF 2017, 'Curated human hyperbilirubinemia data and the respective OATP1B1 and 1B3 inhibition predictions', Data in Brief, vol. 11, pp. 204-207. https://doi.org/10.1016/j.dib.2017.02.009
Showing entries 71 - 80 out of 260